British Dragon Mesterolone Tablets 100 tabs (25 mg/tab) EXPIRATION

Mesterolone – Proviron

Proviron, known for its anti-estrogenic properties, acts by inhibiting estrogen receptors in the brain, thereby stimulating the release of Gonadotropins (LH and FSH), which subsequently prompts the testes to produce more testosterone. This compound does not exhibit direct anabolic or androgenic effects.

Originally synthesized in the 1970s, Proviron disappeared from the market by the late 1990s, with Schering no longer manufacturing it. Online sellers claiming to offer Proviron may be deceptive, and it is likely they are peddling counterfeit items. The drug is mostly believed to be smuggled from Asia, Russia, and Mexico, casting doubt on the authenticity of available products.

Proviron was initially evaluated for treating depression and anxiety in both genders, leading to discoveries that it increased Gonadotropins (LH & FSH) and elevated testosterone levels, which laid the groundwork for its use in fertility issues. However, it is no longer utilized for any medical condition, and the current online offerings are likely not genuine Proviron, but rather fakes or counterfeits.

Indications

Historically, Proviron was prescribed for treating testosterone deficiency and male infertility stemming from issues in the hypothalamus, pituitary, or testes.

Pharmacology

Proviron displays more androgenic than anabolic effects, making it a choice among athletes and bodybuilders recovering from testosterone suppression due to prolonged use of exogenous anabolic steroids. However, many bodybuilders express disappointment, as it often fails to enhance muscle mass or strength, with users frequently deeming it ineffective. The prevalence of counterfeit products exacerbates this issue, as authentic Proviron is nearly impossible to acquire without laboratory testing.

This drug possesses anti-estrogen properties akin to Nolvadex or Arimidex, thereby mitigating common side effects like breast enlargement and water retention associated with anabolic steroids. While some users report increased muscle definition, attributing growth to Proviron amidst multiple steroid use clouds the attributions made. Consequently, many athletes have favored Arimidex or Nolvadex over Proviron.

Females

In the past, Proviron has been used by women; however, reports of its efficacy are mixed. Due to its anti-estrogen effects, female users should always consult healthcare professionals during treatment.

Dosage

The suggested dosage for Mesterolone is 25 mg taken orally 2-3 times daily for several months, potentially followed by a maintenance phase. Once administered, Proviron is swiftly absorbed into the bloodstream, exhibiting a prolonged half-life of approximately 12-24 hours and remaining detectable in urine for up to 2 weeks post-administration.

It is often paired with Tamoxifen or Arimidex during the washout phase due to its insufficient anti-estrogen properties.

Side Effects

Though uncommon, Proviron can cause rare side effects, which, though not experienced by everyone, can be unsettling. Possible side effects include:

• painful erections
• loss of libido
• general fatigue
• deepening of voice
• increased hair growth
• acne and oily skin

Contraindications

Proviron is not recommended for:

• children
• pregnant women
• individuals with abnormal liver function
• men with prostate cancer
• those with allergies

Cost

When available, Proviron is expensive. Its quality and purity remain questionable, as it is exclusively found on the black market, primarily smuggled into the US from Mexico and the Far East. A 20 mg pill typically ranges from $3-$4, yet distinguishing fakes is virtually impossible.

Detection

Proviron is banned by most sporting organizations and is routinely tested for in urine. Given its long half-life, it remains detectable for up to 2 weeks following the final dose.

Legal

Possession of Proviron is not illegal; however, most sporting agencies screen for it in urine tests. In the USA, it falls under the control substance act as a schedule 3 drug.

Final Word

Proviron’s relevance is relegated to history, with genuine products largely unavailable. The current market is flooded with likely fake or contaminated offerings. For those seeking body enhancement, alternatives like Arimidex offer a more reliable option.