British Dragon Mesterolone Tablets 100 tabs (25 mg/tab)

Mesterolone – Proviron

Proviron is an anti-estrogenic medication that blocks estrogen receptors in the brain, prompting a notable increase in Gonadotropins (LH and FSH) and subsequently stimulating testosterone production in the testes. It lacks direct anabolic or androgenic effects.

Synthesized in the 1970s, the drug faded from the market by the late 1990s, with its manufacturer, Schering, ceasing production. Current online sellers of Proviron may be untrustworthy, likely offering counterfeit products. While it’s reported that Proviron can be found online, its authenticity remains questionable, as it often appears to be smuggled from locations like Asia, Russia, and Mexico.

Initially tested for use in treating depression and anxiety in both men and women, trials revealed that it increased Gonadotropins (LH & FSH) along with testosterone levels, leading to its application in addressing fertility issues. However, Proviron is no longer clinically available and is not used for any medical conditions, emphasizing that most online offers are likely fake or counterfeit.

Indications

Historically, Proviron was prescribed for testosterone deficiency and male infertility issues due to hypothalamic, pituitary, or testicular dysfunctions.

Pharmacology

This drug exhibits more androgenic than anabolic properties. Athletes and bodybuilders have utilized Proviron for recovery following testosterone suppression from prolonged anabolic steroid use. However, the majority of users report dissatisfaction, claiming no significant gains in muscle mass or strength, possibly due to purchasing counterfeit products. Like Nolvadex or Arimidex, Proviron possesses anti-estrogenic properties, mitigating side effects like breast enlargement and water retention commonly associated with anabolic steroids.

Some users advocate that it promotes muscle definition, though it’s challenging to attribute effects to Proviron, given the concurrent use of other anabolic steroids. Typically, it is employed during washout phases to support testosterone levels; knowledgeable athletes often prefer alternatives like Arimidex or Nolvadex.

Females

In the past, females have also used Proviron. Reports on its bodybuilding effects are mixed, with many women indicating minimal impact. Due to its anti-estrogen properties, female users should be monitored by healthcare professionals.

Dosage

The recommended dosage of Mesterolone is 25 mg taken orally 2-3 times daily for several months, followed by maintenance therapy. Upon oral administration, it is quickly absorbed into the bloodstream and has a prolonged half-life of 12-24 hours, remaining detectable in urine for at least 2 weeks post-dose.

As an ineffective anti-estrogen, it is commonly combined with Tamoxifen or Arimidex during washout phases.

Side effects

Proviron can lead to rare side effects, which may include:

• painful erections
• diminished libido
• general fatigue
• voice deepening
• increased hair growth
• acne and oily skin

Contraindications

This drug is not advisable for:

• children
• pregnant women
• individuals with liver dysfunction
• those with prostate cancer
• individuals with allergies

Cost

When obtainable, Proviron is costly, with quality and purity in question. Currently, all availability is on the black market, primarily smuggled into the US from Mexico and the Far East, costing about $3-$4 per 20 mg pill, raising concerns about authenticity.

Detection

Proviron is a banned substance in most sports organizations and is actively tested for in urine, remaining detectable for up to 2 weeks due to its lengthy half-life.

Legal

Possession of Proviron is not illegal; however, sporting agencies monitor for its presence in urine tests. In the United States, it is classified as a Schedule III controlled substance.

Final Word

Proviron has become a relic of the past. Genuine products are no longer available, and what is currently on offer is likely counterfeit or contaminated. For those aiming to enhance body performance, alternatives such as Arimidex are recommended.